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Esther Roehn-Carnemolla
Esther Roehn-Carnemolla
Novartis
Biochemistry
Tricyclic
Chemistry
Stereochemistry
Organic chemistry
2
Papers
24
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Identification and optimisation of 4,5-dihydrobenzo[1,2-d:3,4-d]bisthiazole and 4,5-dihydrothiazolo[4,5-h]quinazoline series of selective phosphatidylinositol-3 kinase alpha inhibitors
2015
Bioorganic & Medicinal Chemistry Letters
Robin Alec Fairhurst
Marc Gerspacher
Patricia Imbach-Weese
Robert Mah
Giorgio Caravatti
Pascal Furet
Christine Fritsch
Christian Schnell
Joachim Blanz
Francesca Blasco
Sandrine Desrayaud
Daniel Guthy
Mark Knapp
Dorothee Arz
Jasmin Wirth
Esther Roehn-Carnemolla
Van Huy Luu
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Citations (11)
Discovery of a novel tricyclic 4H-thiazolo[5′,4′:4,5]pyrano[2,3-c]pyridine-2-amino scaffold and its application in a PI3Kα inhibitor with high PI3K isoform selectivity and potent cellular activity
2015
Bioorganic & Medicinal Chemistry Letters
Marc Gerspacher
Robin Alec Fairhurst
Robert Mah
Esther Roehn-Carnemolla
Pascal Furet
Christine Fritsch
Daniel Guthy
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Citations (13)
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