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Stefan Westin
Stefan Westin
Exelixis
Nuclear receptor
Farnesoid X receptor
Biology
Biochemistry
G protein-coupled bile acid receptor
5
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959
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0.02
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Discovery of XL335 (WAY-362450), a Highly Potent, Selective, and Orally Active Agonist of the Farnesoid X Receptor (FXR)
2009
Journal of Medicinal Chemistry
Brenton T. Flatt
Richard J. Martin
Tie Lin Wang
Paige Mahaney
Brett Murphy
Xiao-Hui Gu
Paul A. Foster
Jiali Li
Parinaz C. Pircher
Mary Petrowski
Ira G. Schulman
Stefan Westin
Jay Wrobel
Grace Yan
Eric D. Bischoff
Chris L. Daige
Raju Mohan
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Citations (125)
Regulation of complement C3 expression by the bile acid receptor FXR.
2005
Journal of Biological Chemistry
Jiali Li
Parinaz C. Pircher
Ira G. Schulman
Stefan Westin
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Citations (81)
Molecular Determinants of Crosstalk between Nuclear Receptors and Toll-like Receptors
2005
Cell
Sumito Ogawa
Jean Lozach
Christopher Benner
Gabriel Pascual
Rajendra K. Tangirala
Stefan Westin
Alexander Hoffmann
Shankar Subramaniam
Michael David
Michael G. Rosenfeld
Christopher K. Glass
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Citations (581)
FXR, A Therapeutic Target for Bile Acid and Lipid Disorders
2005
Mini-reviews in Medicinal Chemistry
Stefan Westin
Richard A. Heyman
Richard J. Martin
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Citations (21)
Farnesoid X Receptor Regulates Bile Acid-Amino Acid Conjugation
2003
Journal of Biological Chemistry
Parinaz C. Pircher
Jennifer L. Kitto
Mary Petrowski
Rajendra K. Tangirala
Eric D. Bischoff
Ira G. Schulman
Stefan Westin
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Citations (151)
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