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Hideaki Funami
Hideaki Funami
Chemistry
Inverse agonist
Receptor
Ghrelin
Drug Inverse Agonism
3
Papers
11
Citations
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Structural Optimization of Ghrelin Receptor Inverse Agonists to Improve Lipophilicity and Avoid Mechanism-Based CYP3A4 Inactivation
2015
Chemical & Pharmaceutical Bulletin
Bitoku Takahashi
Hideaki Funami
Makoto Shibata
Hiroshi Maruoka
Makoto Koyama
Satomi Kanki
Tsuyoshi Muto
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Citations (1)
Orally active ghrelin receptor inverse agonists and their actions on a rat obesity model
2015
Bioorganic & Medicinal Chemistry
Bitoku Takahashi
Hideaki Funami
Takehiko Iwaki
Hiroshi Maruoka
Makoto Shibata
Makoto Koyama
Asako Nagahira
Yoshiyuki Kamiide
Satomi Kanki
Yoshiyuki Igawa
Tsuyoshi Muto
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Citations (7)
2-Aminoalkyl nicotinamide derivatives as pure inverse agonists of the ghrelin receptor
2015
Bioorganic & Medicinal Chemistry Letters
Bitoku Takahashi
Hideaki Funami
Takehiko Iwaki
Hiroshi Maruoka
Asako Nagahira
Makoto Koyama
Yoshiyuki Kamiide
Tsuyoshi Matsuo
Tsuyoshi Muto
Hirokazu Annoura
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Citations (3)
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