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Brian Chamberlain
Brian Chamberlain
Cubist Pharmaceuticals
Chemistry
Immunology
Ulcerative colitis
CCR9
Chemokine receptor
4
Papers
24
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Abstract LB-A20: True small molecule STING agonist generates systemic and potent anti-tumor immunity required for effective cancer immunotherapy
2019
Molecular Cancer Therapeutics
Meghana M. Kulkarni
Timothy Dwight
Kristen Marino
Bryce K. Allen
Mohammed Taimi
Cecilia Bastos
Sujen Lai
Cheryl Koh
Ramya Samant
Bethany Tesar
Huang Huang
Brian Chamberlain
James M. Rice
Dazhi Tan
Zhixiong Lin
Sharon Shechter
Stella Li
Sam Sparks
Holly Soutter
Steven Swann
Woody Sherman
Christopher Winter
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Discovery of indole inhibitors of chemokine receptor 9 (CCR9).
2016
Bioorganic & Medicinal Chemistry Letters
Bhaumik A. Pandya
Christian Baber
Audrey Chan
Brian Chamberlain
Haoqun Chandonnet
Jennifer Goss
Timothy Hopper
Blaise Lippa
Katherine M. Poutsiaka
Jan Romero
Sabrina Stucka
Mustafa Varoglu
Jing Zhang
Xin Zhang
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Discovery of Azaindole Ureas as a Novel Class of Bacterial Gyrase B Inhibitors.
2015
Journal of Medicinal Chemistry
Jing Zhang
Qingyi Yang
Jason B. Cross
Jan Antoinette C. Romero
Katherine M. Poutsiaka
Felix Epie
Douglas E. Bevan
Bin Wang
Yanzhi Zhang
Ajit Chavan
Xin Zhang
Terence Moy
Anu Daniel
Kien Nguyen
Brian Chamberlain
Nicole Carter
Joseph Shotwell
Jared Silverman
Chester A. Metcalf
Dominic Ryan
Blaise Lippa
Roland E. Dolle
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Citations (16)
Biarylsulfonamide CCR9 inhibitors for inflammatory bowel disease.
2015
Bioorganic & Medicinal Chemistry Letters
Jing Zhang
Jan Romero
Audrey Chan
Jennifer Goss
Sabrina Stucka
Jason B. Cross
Brian Chamberlain
Mustafa Varoglu
Haoqun Chandonnet
Dominic Ryan
Blaise Lippa
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Citations (8)
1