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Johannes Pilakowski
Johannes Pilakowski
Technische Universität Darmstadt
Chemistry
Zebrafish
Glycogen synthase
Oxadiazole
Biochemistry
3
Papers
32
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Illuminating a Dark Kinase: Structure-Guided Design, Synthesis, and Evaluation of a Potent Nek1 Inhibitor and Its Effects on the Embryonic Zebrafish Pronephros
2021
Journal of Medicinal Chemistry
Georg Baumann
Tobias Meckel
Kevin Böhm
Yung-Hsin Shih
Mirco Dickhaut
Torben Reichardt
Johannes Pilakowski
Ulrich Pehl
Boris Schmidt
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Design, synthesis and biological evaluation of novel aminopyrazole- and 7-azaindole-based Nek1 inhibitors and their effects on zebrafish kidney development.
2021
Bioorganic & Medicinal Chemistry Letters
Johannes Pilakowski
Georg Baumann
Yung-Hsin Shih
Tobias Meckel
Boris Schmidt
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Structure-based optimization of oxadiazole-based GSK-3 inhibitors
2013
European Journal of Medicinal Chemistry
Fabio Lo Monte
T. H. Kramer
Jiamin Gu
Martin Brodrecht
Johannes Pilakowski
Ana Fuertes
Juan Manuel Dominguez
Batya Plotkin
Hagit Eldar-Finkelman
Boris Schmidt
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Citations (30)
1