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Mayuko Akiu
Mayuko Akiu
Daiichi Sankyo
Chemistry
Nucleotide salvage
Nicotinamide phosphoribosyltransferase
Activator (genetics)
NAD+ kinase
4
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5
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0
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2024
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Discovery of DS68702229 as a Potent, Orally Available NAMPT (Nicotinamide Phosphoribosyltransferase) Activator.
2021
Chemical & Pharmaceutical Bulletin
Mayuko Akiu
Takashi Tsuji
Kouki Iida
Yoshitaka Sogawa
Koji Terayama
Mika Yokoyama
Jun Tanaka
Daigo Asano
Tomohiro Honda
Ken Sakurai
Anthony B. Pinkerton
Tsuyoshi Nakamura
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Discovery of 1-[2-(1-methyl-1H-pyrazol-5-yl)-[1,2,4]triazolo[1,5-a]pyridin-6-yl]-3-(pyridin-4-ylmethyl)urea as a potent NAMPT (nicotinamide phosphoribosyltransferase) activator with attenuated CYP inhibition.
2021
Bioorganic & Medicinal Chemistry Letters
Mayuko Akiu
Takashi Tsuji
Yoshitaka Sogawa
Koji Terayama
Mika Yokoyama
Jun Tanaka
Daigo Asano
Ken Sakurai
Eduard Sergienko
E. Hampton Sessions
Stephen J. Gardell
Anthony B. Pinkerton
Tsuyoshi Nakamura
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Optimization of a Urea-containing Series of Nicotinamide Phosphoribosyltransferase (NAMPT) Activators.
2021
Bioorganic & Medicinal Chemistry Letters
Anthony B. Pinkerton
E. Hampton Sessions
Paul Hershberger
Patrick R. Maloney
Satyamaheshwar Peddibhotla
Meghan E. Hopf
Eduard Sergienko
Chen-Ting Ma
Layton H. Smith
Michael R. Jackson
Jun Tanaka
Takashi Tsuji
Mayuko Akiu
Steven E. Cohen
Tsuyoshi Nakamura
Stephen J. Gardell
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Synthesis and biological evaluation of novel imidazol-1-ylacetic acid derivatives as non-brain penetrant bombesin receptor subtype-3 (BRS-3) agonists.
2016
Bioorganic & Medicinal Chemistry Letters
Yohei Kiyotsuka
Kousei Shimada
Shozo Kobayashi
Masanori Suzuki
Mayuko Akiu
Masayoshi Asano
Yoshitaka Sogawa
Takashi Hara
Masahiro Konishi
Rie Abe-Ohya
Masanori Izumi
Yoko Nagai
Kazuhiro Yoshida
Yasuyuki Abe
Hideo Takamori
Hisashi Takahashi
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Citations (4)
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