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Giovanni Cambi
Giovanni Cambi
University of Florence
Ligand
Chemistry
Chemical synthesis
GABAA receptor
Stereochemistry
4
Papers
56
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Structural Constraint at 3-Position of Pirazolo[1,5-a]Pyrimidines as TSPO Ligands Useful for PET-Imaging of Central Nervous System Disease
2009
Chiara Guarino
Giovanni Cambi
Silvia Selleri
Fabrizio Bruni
Gabriella Guerrini
Giovanna Ciciani
Annarella Costanzo
Eleonora Da Pozzo
Claudia Martini
Michael Kassiou
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Synthesis, in Vivo Evaluation, and Molecular Modeling Studies of New Pyrazolo[5,1-c][1,2,4]benzotriazine 5-Oxide Derivatives. Identification of a Bifunctional Hydrogen Bond Area Related to the Inverse Agonism
2009
Journal of Medicinal Chemistry
Gabriella Guerrini
Giovanna Ciciani
Giovanni Cambi
Fabrizio Bruni
Silvia Selleri
Chiara Guarino
Fabrizio Melani
Marina Montali
Claudia Martini
Carla Ghelardini
Monica Norcini
Annarella Costanzo
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Citations (18)
Novel 3-aroylpyrazolo[5,1-c][1,2,4]benzotriazine 5-oxides 8-substituted, ligands at GABAA/benzodiazepine receptor complex: synthesis, pharmacological and molecular modeling studies.
2008
Bioorganic & Medicinal Chemistry
Gabriella Guerrini
Giovanna Ciciani
Giovanni Cambi
Fabrizio Bruni
Silvia Selleri
Fabrizio Melani
Marina Montali
Claudia Martini
Carla Ghelardini
Monica Norcini
Annarella Costanzo
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Novel 3 -iodo -8 -ethoxypyrazolo [5,1-c][1,2,4 ]benzotriazine 5-oxide as promising lead for design of α5-inverse agonist useful tools for therapy of mnemonic damage
2007
Bioorganic & Medicinal Chemistry
Gabriella Guerrini
Giovanna Ciciani
Giovanni Cambi
Fabrizio Bruni
Silvia Selleri
François Besnard
Marina Montali
Claudia Martini
Carla Ghelardini
Nicoletta Galeotti
Annarella Costanzo
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Citations (16)
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