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Megan M. Breiner
Megan M. Breiner
Vanderbilt University
Biochemistry
Chemistry
Stereochemistry
In vivo
Potency
3
Papers
41
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Discovery of Novel Central Nervous System Penetrant Metabotropic Glutamate Receptor Subtype 2 (mGlu2) Negative Allosteric Modulators (NAMs) Based on Functionalized Pyrazolo[1,5-a]pyrimidine-5-carboxamide and Thieno[3,2-b]pyridine-5-carboxamide Cores
2019
Journal of Medicinal Chemistry
Elizabeth S. Childress
Joshua M. Wieting
Andrew S. Felts
Megan M. Breiner
Madeline F. Long
Vincent B. Luscombe
Alice L. Rodriguez
Hyekyung P. Cho
Anna L. Blobaum
Colleen M. Niswender
Kyle A. Emmitte
P. Jeffrey Conn
Craig W. Lindsley
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Citations (10)
Discovery and characterization of N-(1,3-dialkyl-1H-indazol-6-yl)-1H-pyrazolo[4,3-b]pyridin-3-amine scaffold as mGlu4 positive allosteric modulators that mitigate CYP1A2 induction liability
2018
Bioorganic & Medicinal Chemistry Letters
Darren W. Engers
Sean R. Bollinger
Julie L. Engers
Joseph D. Panarese
Megan M. Breiner
Alison R. Gregro
Anna L. Blobaum
Joanne J. Bronson
Yong-Jin Wu
John E. Macor
Alice L. Rodriguez
Rocio Zamorano
P. Jeffrey Conn
Craig W. Lindsley
Colleen M. Niswender
Corey R. Hopkins
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Citations (7)
Design and synthesis of N-aryl phenoxyethoxy pyridinones as highly selective and CNS penetrant mGlu3 NAMs
2017
ACS Medicinal Chemistry Letters
Julie L. Engers
Katrina A. Bollinger
Rebecca L. Weiner
Alice L. Rodriguez
Madeline F. Long
Megan M. Breiner
Sichen Chang
Sean R. Bollinger
Michael Bubser
Carrie K. Jones
Ryan D. Morrison
Thomas M. Bridges
Blobaum Al
Colleen M. Niswender
P. Jeffrey Conn
Kyle A. Emmitte
Craig W. Lindsley
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Citations (24)
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