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H. Tanji
H. Tanji
University of Tokyo
Biochemistry
TLR8
Toll-like receptor
Chemistry
Cell culture
4
Papers
102
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Tetrasubstituted imidazoles as incognito Toll-like receptor 8 a(nta)gonists.
2021
Nature Communications
Yi Yang
Adam Csakai
Shuangshuang Jiang
Christina Smith
H. Tanji
Jian Huang
Torey Jones
Kentaro Sakaniwa
Lindsey J. Broadwell
Chengrui Shi
Subada Soti
Umeharu Ohto
Yaohui Fang
Shu Shen
Fei Deng
Toshiyuki Shimizu
Hang Yin
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Citations (2)
Rationally designed small-molecule inhibitors targeting an unconventional pocket on the TLR8 protein-protein interface.
2020
Journal of Medicinal Chemistry
Shuangshuang Jiang
H. Tanji
Kejun Yin
Shuting Zhang
Kentaro Sakaniwa
Jian Huang
Yi Yang
Jing Li
Umeharu Ohto
Toshiyuki Shimizu
Hang Yin
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Citations (9)
Small-molecule inhibition of TLR8 through stabilization of its resting state
2018
Nature Chemical Biology
Shuting Zhang
Zhenyi Hu
H. Tanji
Shuangshuang Jiang
Nabanita Das
Jing Li
Kentaro Sakaniwa
Jin Jin
Yanyan Bian
Umeharu Ohto
Toshiyuki Shimizu
Hang Yin
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Citations (64)
Identification of a Human Toll-Like Receptor (TLR) 8-Specific Agonist and a Functional Pan-TLR Inhibitor in 2-Aminoimidazoles
2016
Journal of Medicinal Chemistry
Mallesh Beesu
Giuseppe Caruso
Alex C. D. Salyer
Nijunj M. Shukla
Karishma K. Khetani
Luke J. Smith
Lauren M. Fox
H. Tanji
Umeharu Ohto
Toshiyuki Shimizu
Sunil A. David
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Citations (27)
1