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Kevin Guertin
Kevin Guertin
Biogen Idec
Interleukin 17
Biology
Gene expression
Biochemistry
Inverse agonist
4
Papers
93
Citations
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MetAP2 Inhibition Modifies Hemoglobin S (HbS) to Delay Polymerization and Improve Blood Flow in Sickle Cell Disease
2019
Blood
Mélanie Demers
Sarah Sturtevant
Kevin Guertin
Dipti Gupta
Kunal Desai
Benjamin Vieira
Alexandra Hicks
Ayman Ismail
Yukio Nakamura
Bronner P. Gonçalves
Giuseppe Di Caprio
Ethan Schonbrun
Scott Hansen
Martin K. Safo
David K. Wood
John M. Higgins
David R. Light
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Citations (1)
Small molecule mediated inhibition of RORγ-dependent gene expression and autoimmune disease pathology in vivo.
2016
Immunology
Daliya Banerjee
Linlin Zhao
Lan Wu
Arumugam Palanichamy
Ayla Ergun
Liaomin Peng
Catherine Quigley
Stefan Hamann
Robert Dunstan
Patrick Cullen
Norm Allaire
Kevin Guertin
Tao Wang
Jianhua Chao
Christine Loh
Jason D. Fontenot
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Citations (42)
Discovery of novel pyrazole-containing benzamides as potent RORγ inverse agonists
2015
Bioorganic & Medicinal Chemistry Letters
Tao Wang
Daliya Banerjee
Tonika Bohnert
Jianhua Chao
Istvan Enyedy
Jason D. Fontenot
Kevin Guertin
Howard Jones
Edward Yin-Shiang Lin
Douglas Marcotte
Tina Talreja
Kurt Van Vloten
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Citations (22)
Discovery of biaryl carboxylamides as potent RORγ inverse agonists
2015
Bioorganic & Medicinal Chemistry Letters
Jianhua Chao
Istvan Enyedy
Kurt Van Vloten
Douglas Marcotte
Kevin Guertin
Richard H. Hutchings
Noel Powell
Howard Jones
Tonika Bohnert
Chi-Chi Peng
Laura Silvian
Victor Hong
Kevin Little
Daliya Banerjee
Liaomin Peng
Arthur G. Taveras
Joanne L. Viney
Jason D. Fontenot
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Citations (28)
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