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Anne Mengel
Anne Mengel
Bayer
Chemistry
Cancer research
Kinase
BUB1
TANK-binding kinase 1
4
Papers
32
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Discovery of BAY-985 a highly selective TBK1/Ikkε inhibitor
2020
Journal of Medicinal Chemistry
Julien Lefranc
Volker Schulze
R.C. Hillig
Hans Briem
Florian Prinz
Anne Mengel
Tobias Heinrich
Jozsef Bálint
Srinivasan Rengachari
Horst Irlbacher
Detlef Stöckigt
Ulf Bömer
Benjamin Bader
Stefan Gradl
Carl Friedrich Nising
Franz von Nussbaum
Dominik Mumberg
Daniel Panne
Antje Margret Wengner
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Discovery of BAY-985, a Highly Selective TBK1/IKKε Inhibitor.
2020
Journal of Medicinal Chemistry
Julien Lefranc
V.K. Schulze
R.C. Hillig
Hans Briem
Florian Prinz
Anne Mengel
Tobias Heinrich
József Bálint
Srinivasan Rengachari
Horst Irlbacher
Detlef Stöckigt
Ulf Bömer
Benjamin Bader
Stefan Gradl
Carl Friedrich Nising
Franz von Nussbaum
Dominik Mumberg
Daniel Panne
Antje Margret Wengner
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Citations (10)
Inhibition of BUB1 Kinase by BAY 1816032 Sensitizes Tumor Cells toward Taxanes, ATR, and PARP Inhibitors In Vitro and In Vivo
2019
Clinical Cancer Research
Gerhard Siemeister
Anne Mengel
Amaury E. Fernández-Montalván
Wilhelm Bone
Jens Schröder
Sabine Zitzmann-Kolbe
Hans Briem
Stefan Prechtl
Simon Holton
Ursula Mönning
Oliver von Ahsen
Sandra Johanssen
Arwed Cleve
Vera Pütter
Marion Hitchcock
Franz von Nussbaum
Michael Brands
Karl Ziegelbauer
Dominik Mumberg
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Citations (22)
Crystal structure of the human Bub1 kinase domain in complex with BAY 1816032
2018
Simon Holton
Gerhard Siemeister
Anne Mengel
Wilhelm Bone
J. Schroeder
Sabine Zitzmann-Kolbe
Hans Briem
Amaury E. Fernández-Montalván
Stefan Prechtl
Ursula Moenning
O von Ahsen
J. Johanssen
Arwed Cleve
Vera Puetter
Marion Hitchcock
F. von Nussbaum
Michael Brands
Dominik Mumberg
Karl Ziegelbauer
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