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Tomoshige Numazawa
Tomoshige Numazawa
Merck & Co.
Biochemistry
Chemistry
Muscarinic acetylcholine receptor
Muscarinic acetylcholine receptor M2
Receptor
2
Papers
39
Citations
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Pharmacological Properties of (2R)-N-[1-(6-Aminopyridin-2-ylmethyl)piperidin-4-yl]-2-[(1R)-3,3-difluorocyclopentyl]-2- hydroxy-2-phenylacetamide: A Novel Muscarinic Antagonist with M2-Sparing Antagonistic Activity
2001
Journal of Pharmacology and Experimental Therapeutics
Hiroyasu Hirose
Ikuo Aoki
Toshifumi Kimura
Toru Fujikawa
Tomoshige Numazawa
Kaori Sasaki
Akio Sato
Takuro Hasegawa
Masaru Nishikibe
Morihiro Mitsuya
Norikazu Ohtake
Toshiaki Mase
Kazuhito Noguchi
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Citations (21)
Discovery of a muscarinic M3 receptor antagonist with high selectivity for M3 over M2 receptors among 2-[(1S,3S)-3-sulfonylaminocyclopentyl]phenylacetamide derivatives
2000
Bioorganic & Medicinal Chemistry
Morihiro Mitsuya
Yoshio Ogino
Kumiko Kawakami
Minaho Uchiyama
Toshifumi Kimura
Tomoshige Numazawa
Takuro Hasegawa
Norikazu Ohtake
Kazuhito Noguchi
Toshiaki Mase
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Citations (18)
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