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Christopher J. Brassard
Christopher J. Brassard
Vanderbilt University
Biochemistry
Potency
Chemistry
Pharmacophore
Aldehyde oxidase
2
Papers
23
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Discovery of 4-alkoxy-6-methylpicolinamide negative allosteric modulators of metabotropic glutamate receptor subtype 5
2019
Bioorganic & Medicinal Chemistry Letters
Andrew S. Felts
Katrina A. Bollinger
Christopher J. Brassard
Alice L. Rodriguez
Ryan D. Morrison
J. Scott Daniels
Anna L. Blobaum
Colleen M. Niswender
Carrie K. Jones
P. Jeffrey Conn
Kyle A. Emmitte
Craig W. Lindsley
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Design and Synthesis of mGlu2 NAMs with Improved Potency and CNS Penetration Based on a Truncated Picolinamide Core
2017
ACS Medicinal Chemistry Letters
Katrina A. Bollinger
Andrew S. Felts
Christopher J. Brassard
Julie L. Engers
Alice L. Rodriguez
Rebecca L. Weiner
Hyekyung P. Cho
Sichen Chang
Michael Bubser
Carrie K. Jones
Anna L. Blobaum
Colleen M. Niswender
P. Jeffrey Conn
Kyle A. Emmitte
Craig W. Lindsley
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Citations (20)
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