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Marina Bukhtiyarova

14

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297

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Synthesis and pharmacological evaluation of N-(3-(1H-indol-4-yl)-5-(2-methoxyisonicotinoyl)phenyl)methanesulfonamide (LP-261), a potent antimitotic agent.

2011 Journal of Medicinal Chemistry
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The rational design of a novel potent analogue of the 5’-AMP-activated protein kinase inhibitor compound C with improved selectivity and cellular activity

2010 Bioorganic & Medicinal Chemistry Letters
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protein kinase inhibitor compound C with improved selectivity and cellular activity

2010
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Discovery and SAR of a series of 4,6-diamino-1,3,5-triazin-2-ol as novel non-nucleoside reverse transcriptase inhibitors of HIV-1.

2010 Bioorganic & Medicinal Chemistry Letters
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Analysis of imatinib and sorafenib binding to p38alpha compared with c-Abl and b-Raf provides structural insights for understanding the selectivity of inhibitors targeting the DFG-out form of protein kinases.

2010 Biochemistry
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Conformational plasticity of p38 MAP kinase DFG motif mutants in response to inhibitor binding

2010
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Structure-based design of substituted biphenyl ethylene ethers as ligands binding in the hydrophobic pocket of gp41 and blocking the helical bundle formation.

2009 Bioorganic & Medicinal Chemistry Letters
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Crystal Structure of F169R p38 Kinase

2007
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Mutagenesis of p38alpha MAP kinase establishes key roles of Phe169 in function and structural dynamics and reveals a novel DFG-OUT state.

2007 Biochemistry
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Crystal Structure of F169A p38 Kinase

2007
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