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Natasja M.W.J. de Bruin
Natasja M.W.J. de Bruin
Solvay
Biochemistry
Chemistry
Pyrazoline
Organic chemistry
Receptor
3
Papers
59
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Optimization of N′-(arylsulfonyl)pyrazoline-1-carboxamidines by exploiting a novel interaction site in the 5-HT6 antagonistic binding pocket
2016
Bioorganic & Medicinal Chemistry Letters
Arnold van Loevezijn
J. Venhorst
Wouter I. Iwema-Bakker
Jos H.M. Lange
Wouter de Looff
Remco Henzen
Jelle de Vries
Rob P. van de Woestijne
Arnold P. den Hartog
Stefan Verhoog
Martina A.W. van der Neut
Natasja M.W.J. de Bruin
Chris G. Kruse
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Citations (3)
N′-(Arylsulfonyl)pyrazoline-1-carboxamidines as Novel, Neutral 5-Hydroxytryptamine 6 Receptor (5-HT6R) Antagonists with Unique Structural Features
2011
Journal of Medicinal Chemistry
Arnold van Loevezijn
Jennifer Venhorst
Wouter I. Iwema-Bakker
Cor G. de Korte
Wouter de Looff
Stefan Verhoog
Jan-Willem van Wees
Martijn van Hoeve
Rob P. van de Woestijne
Martina A.W. van der Neut
Alice J.M. Borst
Maria J.P. Van Dongen
Natasja M.W.J. de Bruin
Hiskias G. Keizer
Chris G. Kruse
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Citations (35)
Biophysical and physicochemical methods differentiate highly ligand-efficient human D-amino acid oxidase inhibitors
2011
European Journal of Medicinal Chemistry
Jos H.M. Lange
J. Venhorst
Maria J.P. Van Dongen
Jurjen Frankena
Firas Bassissi
Natasja M.W.J. de Bruin
Cathaline den Besten
Stephanie B.A. de Beer
Chris Oostenbrink
Natalia Markova
Chris G. Kruse
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Citations (21)
1