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Akihiro Tasaka

Takeda Pharmaceutical Company

63

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Synthesis and biological evaluation of novel selective androgen receptor modulators (SARMs). Part I

2015 Bioorganic & Medicinal Chemistry
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Effect of a novel 17,20-lyase inhibitor, orteronel (TAK-700), on androgen synthesis in male rats

2013 The Journal of Steroid Biochemistry and Molecular Biology
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Effect of an investigational CYP17A1 inhibitor, orteronel (TAK-700), on estrogen- and corticoid-synthesis pathways in hypophysectomized female rats and on the serum estradiol levels in female cynomolgus monkeys

2013 The Journal of Steroid Biochemistry and Molecular Biology
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Design, synthesis, and biological evaluation of 4-phenylpyrrole derivatives as novel androgen receptor antagonists

2012 Bioorganic & Medicinal Chemistry
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298 Effect of Investigational Agent Orteronel (TAK-700) On Estrogen- and Corticoid-synthesis Pathways in Hypophysectomized Female Rats and On Serum Estradiol in Female Cynomolgus Monkeys

2012 European Journal of Cancer
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Orteronel (TAK-700), a novel non-steroidal 17,20-lyase inhibitor: effects on steroid synthesis in human and monkey adrenal cells and serum steroid levels in cynomolgus monkeys.

2012 The Journal of Steroid Biochemistry and Molecular Biology
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163 Effect of a novel, investigational 17,20-lyase inhibitor, TAK-700, on enzyme activity and serum androgen levels in human H295R cells and cynomolgus monkeys

2010 Ejc Supplements
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Optically Active Antifungal Azoles. Part 6. Synthesis and Antifungal Activity of N-((1R,2R)-2-(2,4-Difluorophenyl)-2-hydroxy-1-methyl-3-(1H- 1,2,4-triazol-1-yl)propyl)-N′-(4-substituted phenyl)-3(2H,4H)-1,2,4- triazolones and 5(1H,4H)

2010 ChemInform
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167 Effects of a novel, investigational 17,20-lyase inhibitor, TAK-700, on androgen synthesis in male rats: in vivo and in vitro specificity studies

2010 Ejc Supplements
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Optically Active Antifungal Azoles. Part 7. Synthesis and Antifungal Activity of Stereoisomers of 2-((1R,2R)-2-(2,4-Difluorophenyl)-2- hydroxy-1-methyl-3-(1H-1,2,4-triazol-1-yl)propyl)-4-(4-(2,2,3,3- tetrafluoropropoxy)phenyl)-3(2H,4H

2010 ChemInform
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