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Rebecca Cowling

15

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Acylguanidine inhibitors of β-secretase : Optimization of the pyrrole ring substituents extending into the S1 and S3 substrate binding pockets

2008 Bioorganic & Medicinal Chemistry Letters
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Thiophene substituted acylguanidines as BACE1 inhibitors.

2007 Bioorganic & Medicinal Chemistry Letters
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A novel approach to identifying β-secretase inhibitors : Bis-statine peptide mimetics discovered using structure and spot synthesis

2006 Peptides
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Acylguanidines as Small-Molecule β-Secretase Inhibitors

2006 Journal of Medicinal Chemistry
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Characterization of (2R, 3S)-2-({[4-(2-butynyloxy)phenyl]sulfonyl}amino)-N,3-dihydroxybutanamide, a potent and selective inhibitor of TNF-α converting enzyme

2004 International Immunopharmacology
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Evaluation of fluorescence-based thermal shift assays for hit identification in drug discovery

2004 Analytical Biochemistry
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Synthesis and SAR of bis-statine based peptides as BACE 1 inhibitors.

2004 Bioorganic & Medicinal Chemistry Letters
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Synthesis and structure-activity relationship of N-substituted 4-arylsulfonylpiperidine-4-hydroxamic acids as novel, orally active matrix metalloproteinase inhibitors for the treatment of osteoarthritis

2003 Journal of Medicinal Chemistry
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Thiomorpholine sulfonamide hydroxamic acid-based TACE inhibitors

2003
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Synthesis and Structure−Activity Relationship of α-Sulfonylhydroxamic Acids as Novel, Orally Active Matrix Metalloproteinase Inhibitors for the Treatment of Osteoarthritis

2003 Journal of Medicinal Chemistry
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Citations (51)