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Tetsuya Tamura
Tetsuya Tamura
Pfizer
Chemistry
Organic chemistry
Biochemistry
Stereochemistry
Imidazole
5
Papers
127
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Synthesis of benzamide derivatives as TRPV1 antagonists.
2008
Bioorganic & Medicinal Chemistry Letters
Yuji Shishido
Madoka Jinno
Takafumi Ikeda
Fumitaka Ito
Masaki Sudo
Naoya Makita
Atsuko Ohta
Ayako Iki-Taki
Takashi Ohmi
Yoshihito Kanai
Tetsuya Tamura
Masato Shimojo
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Citations (14)
Pharmacological properties of a novel nociceptin/orphanin FQ receptor agonist, 2-(3,5-dimethylpiperazin-1-yl)-1-[1-(1-methylcyclooctyl) piperidin-4-yl]-1H-benzimidazole, with anxiolytic potential
2008
European Journal of Pharmacology
Akiko Hirao
Aki Imai
Yutaka Sugie
Tetsuya Tamura
Hirohisa Shimokawa
Katsuo Toide
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Citations (17)
Optimization of Imidazole 5-Lipoxygenase Inhibitors and Selection and Synthesis of a Development Candidate
2005
Chemical & Pharmaceutical Bulletin
Takashi Mano
Rodney W. Stevens
Kazuo Ando
Makoto Kawai
Kiyoshi Kawamura
Kazunari Nakao
Yoshiyuki Okumura
Takako Okumura
Minoru Sakakibara
Kimitaka Miyamoto
Tetsuya Tamura
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Citations (20)
4-[5-fluoro-3-[4-(2-methyl-1h-imidazol-1-yl)benzyloxy]phenyl]-3,4,5,6-tetrahydro -2h-pyran-4-carboxamide, an orally active inhibitor of 5-lipoxygenase with improved pharmacokinetic and toxicology characteristics
2004
Journal of Medicinal Chemistry
Takashi Mano
Yoshiyuki Okumura
Minoru Sakakibara
Takako Okumura
Tetsuya Tamura
Kimitaka Miyamoto
Rodney W. Stevens
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Citations (29)
Novel imidazole compounds as a new series of potent, orally active inhibitors of 5-lipoxygenase
2003
Bioorganic & Medicinal Chemistry
Takashi Mano
Rodney W. Stevens
Kazuo Ando
Kazunari Nakao
Yoshiyuki Okumura
Minoru Sakakibara
Takako Okumura
Tetsuya Tamura
Kimitaka Miyamoto
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Citations (47)
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