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Manfred Kraus
Manfred Kraus
AstraZeneca
Immunology
Biology
In vivo
Cancer research
Apoptosis
4
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21
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Concurrent Inhibition of Pim and FLT3 Kinases Enhances Apoptosis of FLT3-ITD Acute Myeloid Leukemia Cells through Increased Mcl-1 Proteasomal Degradation
2018
Clinical Cancer Research
Shivani Kapoor
Karthika Natarajan
Patrick R. Baldwin
Kshama A. Doshi
Rena G. Lapidus
Trevor J. Mathias
Mario Scarpa
Rossana Trotta
Eduardo Davila
Manfred Kraus
Dennis Huszar
Adriana E. Tron
Danilo Perrotti
Maria R. Baer
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Abstract A24: Comprehensive PI3K pathway inhibition through combination of the PI3Kβ/δ inhibitor AZD8186 and the mTORC1/2 inhibitor AZD2014 drives tumor regression in vivo
2015
Molecular Cancer Therapeutics
Urs Hancox
Urszula M. Polanska
Lyndsay Hanson
Rebecca Ellston
Julia Maynard
Manfred Kraus
Jon Owen Curwen
Teresa Klinowska
Lara Ward
Francisco Cruzalegui
Stephen Green
Stefan Symeonides
Kathryn Cronin
Simon T. Barry
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546 The PI3Kbeta/delta inhibitor AZD8186 combines with the dual mTORC1/2 inhibitor AZD2014 to give comprehensive PI3K pathway inhibition and drive tumour regression in vivo
2014
European Journal of Cancer
B. Simon
Urs Hancox
Urszula M. Polanska
Lyndsey Hanson
Phillippa Dudley
Rebecca Ellston
Juliana Maynard
Manfred Kraus
Jon Owen Curwen
Teresa Klinowska
Lara Ward
Francisco Cruzalegui
Stefan Symeonides
Kathryn Cronin
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The Pim Kinase Inhibitor AZD1208 Enhances Apoptosis Induction By Clinically Active FLT3 Inhibitors in FLT3-ITD Acute Myeloid Leukemia Cells in Vitro and in Vivo through Synergistic Downregulation of Mcl-1 and of Bcl-xL
2014
Blood
Karthika Natarajan
Trevor J. Mathias
Kshama A. Doshi
Adriana E. Tron
Manfred Kraus
Rossana Trotta
Danilo Perrotti
Dennis Huszar
Maria R. Baer
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