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Qi-Kun Yin
Qi-Kun Yin
Sun Yat-sen University
Chemistry
Biochemistry
Helicase
DNA damage
Cell biology
4
Papers
76
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Design, Synthesis and Evaluation of New Quinazolinone Derivatives that Inhibit Bloom's Syndrome Protein (BLM) Helicase, Trigger DNA damage at the Telomere Region and Synergize with PARP Inhibitors.
2020
Journal of Medicinal Chemistry
Chen Xi Wang
Zi Lin Zhang
Qi-Kun Yin
Jia-Li Tu
Jia-En Wang
Yao-Hao Xu
Yong Rao
Tian-Miao Ou
Shi-Liang Huang
Ding Li
Honggen Wang
Qingjiang Li
Jia-Heng Tan
Shuo-Bin Chen
Zhi-Shu Huang
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Citations (4)
Discovery of Isaindigotone Derivatives as Novel Bloom’s Syndrome Protein (BLM) Helicase Inhibitors That Disrupt the BLM/DNA Interactions and Regulate the Homologous Recombination Repair
2019
Journal of Medicinal Chemistry
Qi-Kun Yin
Chen-Xi Wang
Yu-Qing Wang
Qian-Liang Guo
Zi-Lin Zhang
Tian-Miao Ou
Shi-Liang Huang
Ding Li
Honggen Wang
Jia-Heng Tan
Shuo-Bin Chen
Zhi-Shu Huang
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Citations (15)
Design, Synthesis, and Evaluation of New Selective NM23-H2 Binders as c-MYC Transcription Inhibitors via Disruption of the NM23-H2/G-Quadruplex Interaction
2017
Journal of Medicinal Chemistry
Yu-Qing Wang
Zhou-Li Huang
Shuo-Bin Chen
Chen-Xi Wang
Chan Shan
Qi-Kun Yin
Tian-Miao Ou
Ding Li
Lian-Quan Gu
Jia-Heng Tan
Zhi-Shu Huang
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Citations (23)
New Disubstituted Quindoline Derivatives Inhibiting Burkitt’s Lymphoma Cell Proliferation by Impeding c-MYC Transcription
2017
Journal of Medicinal Chemistry
Hui-Yun Liu
Ai-Chun Chen
Qi-Kun Yin
Zeng Li
Su-Mei Huang
Gang Du
Jin-Hui He
Li-Peng Zan
Shi-Ke Wang
Yao-Hao Xu
Jia-Heng Tan
Tian-Miao Ou
Ding Li
Lian-Quan Gu
Zhi-Shu Huang
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Citations (34)
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