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Makoto Hamada
Makoto Hamada
Taisho Pharmaceutical Co.
Chemistry
Biochemistry
Structure–activity relationship
Piperidine
Agonist
5
Papers
26
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Synthesis and Structure-Activity Relationship of C-Phenyl D-Glucitol (TP0454614) Derivatives as Selective Sodium-Dependent Glucose Cotransporter 1 (SGLT1) Inhibitors.
2020
Chemical & Pharmaceutical Bulletin
Shoichi Kuroda
Yohei Kobashi
Madoka Kawamura
Kenichi Kawabe
Fumiyasu Shiozawa
Makoto Hamada
Yuki Shimizu
Lisa Okumura-Kitajima
Hiroko Koretsune
Kayo Kimura
Koji Yamamoto
Hiroyuki Kakinuma
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Down-regulation of CYP1A2, CYP2B6, and CYP3A4 in human hepatocytes by prolyl hydroxylase domain 2 inhibitors via hypoxia-inducible factor-α stabilization.
2020
Drug Metabolism and Disposition
Hiroki Takano
Junichi Yamaguchi
Sota Kato
Makoto Hamada
Mika Tada
Hiromi Endo
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Discovery of novel 2-[(4-hydroxy-6-oxo-2,3-dihydro-1 H -pyridine-5-carbonyl)amino]acetic acid derivatives as HIF prolyl hydroxylase inhibitors for treatment of renal anemia
2018
Bioorganic & Medicinal Chemistry Letters
Makoto Hamada
Tetsuo Takayama
Tsuyoshi Shibata
Akira Hiratate
Masato Takahashi
Miyoko Yashiro
Noriko Takayama
Lisa Okumura-Kitajima
Hiroko Koretsune
Hiromitsu Kajiyama
Takumi Naruse
Sota Kato
Hiroki Takano
Hiroyuki Kakinuma
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Citations (4)
Novel 3 H -[1,2,3]triazolo[4,5- c ]pyridine derivatives as GPR119 agonists: Synthesis and structure-activity/solubility relationships
2017
Bioorganic & Medicinal Chemistry
Daisuke Matsuda
Yohei Kobashi
Ayako Mikami
Madoka Kawamura
Fumiyasu Shiozawa
Kenichi Kawabe
Makoto Hamada
Shinichi Nishimoto
Kayo Kimura
Masako Miyoshi
Noriko Takayama
Hiroyuki Kakinuma
Norikazu Ohtake
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Citations (8)
Design and synthesis of 1H-pyrazolo[3,4-c]pyridine derivatives as a novel structural class of potent GPR119 agonists.
2016
Bioorganic & Medicinal Chemistry Letters
Daisuke Matsuda
Yohei Kobashi
Ayako Mikami
Madoka Kawamura
Fumiyasu Shiozawa
Kenichi Kawabe
Makoto Hamada
Koji Oda
Shinichi Nishimoto
Kayo Kimura
Masako Miyoshi
Noriko Takayama
Hiroyuki Kakinuma
Norikazu Ohtake
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Citations (13)
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