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Jerri L. Rook
Jerri L. Rook
Vanderbilt University
In vivo
Chemistry
Penetrant (mechanical, electrical, or structural)
Pharmacology
cns penetration
2
Papers
1
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0
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2024
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Discovery and optimization of a novel CNS penetrant series of mGlu4 PAMs based on a 1,4-thiazepane core with in vivo efficacy in a preclinical Parkinsonian model.
2021
Bioorganic & Medicinal Chemistry Letters
Caitlin N. Kent
Mark G. Fulton
Kaylee J. Stillwell
Jonathan W. Dickerson
Matthew T. Loch
Alice L. Rodriguez
Anna L. Blobaum
Olivier Boutaud
Jerri L. Rook
Colleen M. Niswender
P. Jeffrey Conn
Craig W. Lindsley
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Discovery of “Molecular Switches” within a Series of mGlu5 Allosteric Ligands Driven by a “Magic Methyl” Effect Affording Both PAMs and NAMs with In Vivo Activity, Derived from an M1 PAM Chemotype
2021
Lisa Barbaro
Alice L. Rodriguez
Ashlyn N. Blevins
Jonathan W. Dickerson
Natasha Billard
Olivier Boutaud
Jerri L. Rook
Colleen M. Niswender
P. Jeffrey Conn
Darren W. Engers
Craig W. Lindsley
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