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Yuichiro Kawamoto
Yuichiro Kawamoto
Astellas Pharma
Chemistry
Biochemistry
Pharmacology
Pyrimidine
Fibroblast growth factor receptor 3
3
Papers
16
Citations
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Synthesis and structure-activity relationships of pyrimidine derivatives as potent and orally active FGFR3 inhibitors with both increased systemic exposure and enhanced in vitro potency.
2021
Bioorganic & Medicinal Chemistry
Ikumi Kuriwaki
Minoru Kameda
Kazuhiko Iikubo
Hiroyuki Hisamichi
Yuichiro Kawamoto
Shigetoshi Kikuchi
Hiroyuki Moritomo
Yutaka Kondoh
Tadashi Terasaka
Yasushi Amano
Yukihiro Tateishi
Yuka Echizen
Yoshinori Iwai
Atsushi Noda
Hiroshi Tomiyama
Taisuke Nakazawa
Masaaki Hirano
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Citations (2)
Structure-based drug design of 1,3,5-triazine and pyrimidine derivatives as novel FGFR3 inhibitors with high selectivity over VEGFR2
2020
Bioorganic & Medicinal Chemistry
Ikumi Kuriwaki
Minoru Kameda
Hiroyuki Hisamichi
Shigetoshi Kikuchi
Kazuhiko Iikubo
Yuichiro Kawamoto
Hiroyuki Moritomo
Yutaka Kondoh
Yasushi Amano
Yukihiro Tateishi
Yuka Echizen
Yoshinori Iwai
Atsushi Noda
Hiroshi Tomiyama
Tomoyuki Suzuki
Masaaki Hirano
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Citations (7)
Identification of potent lysophosphatidic acid receptor 5 (LPA5) antagonists as potential analgesic agents
2018
Bioorganic & Medicinal Chemistry
Yuichiro Kawamoto
Ryushi Seo
Nobuhito Murai
Hideki Hiyama
Hiromasa Oka
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Citations (7)
1