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Shigeki Kunikawa
Shigeki Kunikawa
Astellas Pharma
Chemistry
T cell
Biochemistry
In vivo
Pharmacology
5
Papers
25
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Discovery of 2,4-diamino-5-cyanopyrimidine derivatives as protein kinase C theta inhibitors with mitigated time-dependent drug-drug interactions.
2019
Bioorganic & Medicinal Chemistry
Shigeki Kunikawa
Akira Tanaka
Yuji Takasuna
Mamoru Tasaki
Noboru Chida
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Citations (2)
A novel 2,4-diaminopyrimidine derivative as selective inhibitor of protein kinase C theta prevents allograft rejection in a rat heart transplant model
2018
Bioorganic & Medicinal Chemistry
Shigeki Kunikawa
Akira Tanaka
Yuji Takasuna
Mamoru Tasaki
Noboru Chida
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Corrigendum to “Synthesis and evaluation of novel 1H-pyrrolo[2,3-b]pyridine-5-carboxamide derivatives as potent and orally efficacious immunomodulators targeting JAK3” [Bioorg. Med. Chem. 23 (2015) 4871–4883]
2016
Bioorganic & Medicinal Chemistry
Yutaka Nakajima
Takayuki Inoue
Kazuo Nakai
Koichiro Mukoyoshi
Hisao Hamaguchi
Keiko Hatanaka
Hiroshi Sasaki
Akira Tanaka
Fumie Takahashi
Shigeki Kunikawa
Hiroyuki Usuda
Ayako Moritomo
Yasuyuki Higashi
Masamichi Inami
Shohei Shirakami
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Citations (1)
Synthesis and evaluation of novel 1H-pyrrolo[2,3-b]pyridine-5-carboxamide derivatives as potent and orally efficacious immunomodulators targeting JAK3.
2015
Bioorganic & Medicinal Chemistry
Yutaka Nakajima
Takayuki Inoue
Kazuo Nakai
Koichiro Mukoyoshi
Hisao Hamaguchi
Keiko Hatanaka
Hiroshi Sasaki
Akira Tanaka
Fumie Takahashi
Shigeki Kunikawa
Hiroyuki Usuda
Ayako Moritomo
Yasuyuki Higashi
Masamichi Inami
Shohei Shirakami
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Citations (14)
Optimization of 2,4-diamino-5-fluoropyrimidine derivatives as protein kinase C theta inhibitors with mitigated time-dependent drug-drug interactions and P-gp liability.
2015
Bioorganic & Medicinal Chemistry
Shigeki Kunikawa
Akira Tanaka
Koichiro Mukoyoshi
Shinya Nagashima
Hiroaki Tominaga
Noboru Chida
Mamoru Tasaki
Fumiyuki Shirai
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Citations (6)
1