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George Eiermann
George Eiermann
Protein Sciences
Omarigliptin
Dipeptidyl peptidase-4
Biochemistry
Structure–activity relationship
Chemistry
2
Papers
26
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The discovery of novel 5,6,5- and 5,5,6-tricyclic pyrrolidines as potent and selective DPP-4 inhibitors.
2016
Bioorganic & Medicinal Chemistry Letters
Jason M. Cox
Hong D. Chu
Jeffrey T. Kuethe
Ying-Duo Gao
Giovanna Scapin
George Eiermann
Huaibing He
Xiaohua Li
Kathryn A. Lyons
Joseph M. Metzger
Aleksandr Petrov
Joseph K. Wu
Shiyao Xu
Ranabir SinhaRoy
Ann E. Weber
Tesfaye Biftu
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Citations (15)
Structure–activity-relationship of amide and sulfonamide analogs of omarigliptin
2015
Bioorganic & Medicinal Chemistry Letters
Ping Chen
Dennis Feng
Xiaoxia Qian
James M. Apgar
Robert R. Wilkening
Jeffrey T. Kuethe
Ying-Duo Gao
Giovanna Scapin
Jason M. Cox
George A. Doss
George Eiermann
Huaibing He
Xiaohua Li
Kathryn A. Lyons
Joseph M. Metzger
Aleksandr Petrov
Joseph K. Wu
Shiyao Xu
Ann E. Weber
Youwei Yan
Ranabir Sinha Roy
Tesfaye Biftu
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Citations (11)
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