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Craig A. Behnke
Craig A. Behnke
Takeda Pharmaceutical Company
Chemistry
Bioavailability
Stereochemistry
Renin inhibitor
Lead compound
5
Papers
58
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Discovery of benzimidazole derivatives as orally active renin inhibitors: Optimization of 3,5-disubstituted piperidine to improve pharmacokinetic profile.
2018
Bioorganic & Medicinal Chemistry
Hidekazu Tokuhara
Yasuhiro Imaeda
Yoshiyuki Fukase
Koichi Iwanaga
Naohiro Taya
Koji Watanabe
Ray Kanagawa
Keisuke Matsuda
Yumiko Kajimoto
Keiji Kusumoto
Mitsuyo Kondo
Gyorgy Snell
Craig A. Behnke
Takanobu Kuroita
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Citations (4)
Novel approach of fragment-based lead discovery applied to renin inhibitors
2016
Bioorganic & Medicinal Chemistry
Michiko Tawada
Shinkichi Suzuki
Yasuhiro Imaeda
Hideyuki Oki
Gyorgy Snell
Craig A. Behnke
Mitsuyo Kondo
Naoki Tarui
Toshimasa Tanaka
Takanobu Kuroita
Masaki Tomimoto
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Citations (3)
Structure-based design of a new series of N-(piperidin-3-yl)pyrimidine-5-carboxamides as renin inhibitors
2016
Bioorganic & Medicinal Chemistry
Yasuhiro Imaeda
Michiko Tawada
Shinkichi Suzuki
Masaki Tomimoto
Mitsuyo Kondo
Naoki Tarui
Tsukasa Sanada
Ray Kanagawa
Gyorgy Snell
Craig A. Behnke
Keiji Kubo
Takanobu Kuroita
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Citations (6)
Discovery of TAK-272: A Novel, Potent, and Orally Active Renin Inhibitor.
2016
ACS Medicinal Chemistry Letters
Yasuhiro Imaeda
Hidekazu Tokuhara
Yoshiyuki Fukase
Ray Kanagawa
Yumiko Kajimoto
Keiji Kusumoto
Mitsuyo Kondo
Gyorgy Snell
Craig A. Behnke
Takanobu Kuroita
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Citations (18)
Synthesis, SAR study, and biological evaluation of a series of piperazine ureas as fatty acid amide hydrolase (FAAH) inhibitors
2013
Bioorganic & Medicinal Chemistry
Mitsunori Kono
Takahiro Matsumoto
Toru Kawamura
Atsushi Nishimura
Yoshihiro Kiyota
Hideyuki Oki
Junichi Miyazaki
Shigeru Igaki
Craig A. Behnke
Masato Shimojo
Masakuni Kori
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Citations (27)
1