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Richard Thomas Beresis
Richard Thomas Beresis
Neuroactive steroid
GABAA receptor
Aminobutyric acid
Allosteric regulation
Pregnanolone
2
Papers
69
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Neuroactive Steroids. 2. 3α-Hydroxy-3β-methyl-21-(4-cyano-1H-pyrazol-1′-yl)-19-nor-5β-pregnan-20-one (SAGE-217): A Clinical Next Generation Neuroactive Steroid Positive Allosteric Modulator of the (γ-Aminobutyric Acid)A Receptor
2017
Journal of Medicinal Chemistry
Gabriel Martinez-Botella
Francesco G. Salituro
Boyd L. Harrison
Richard Thomas Beresis
Zhu Bai
Maria-Jesus Blanco
Gabriel M. Belfort
Jing Dai
Carlos M. Loya
Michael A. Ackley
Alison L. Althaus
Scott J. Grossman
Ethan Hoffmann
James Doherty
Albert Jean Robichaud
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Citations (44)
Neuroactive Steroids. 1. Positive Allosteric Modulators of the (γ-Aminobutyric Acid)A Receptor: Structure–Activity Relationships of Heterocyclic Substitution at C-21
2015
Journal of Medicinal Chemistry
Gabriel Martinez-Botella
Francesco G. Salituro
Boyd L. Harrison
Richard Thomas Beresis
Zhu Bai
Kaisheng Shen
Gabriel M. Belfort
Carlos M. Loya
Michael A. Ackley
Scott J. Grossman
Ethan Hoffmann
Shiling Jia
Jiamiao Wang
James Doherty
Albert Jean Robichaud
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Citations (25)
1