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Hiroyasu Tsuge
Hiroyasu Tsuge
Merck & Co.
Neuropeptide Y receptor
Biochemistry
Chemistry
Antagonist
Chemical synthesis
3
Papers
45
Citations
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Novel orally active NPY Y5 receptor antagonists: Synthesis and structure–activity relationship of spiroindoline class compounds
2009
Bioorganic & Medicinal Chemistry
Toshihiro Sakamoto
Minoru Moriya
Hiroyasu Tsuge
Toshiyuki Takahashi
Yuji Haga
Katsumasa Nonoshita
Osamu Okamoto
Hirobumi Takahashi
Aya Sakuraba
Tomoko Hirohashi
Takunobu Shibata
Tetsuya Kanno
Junko Ito
Hisashi Iwaasa
Akira Gomori
Akane Ishihara
Takahiro Fukuroda
Akio Kanatani
Takehiro Fukami
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Citations (10)
Discovery of tetrasubstituted imidazolines as potent and selective neuropeptide Y Y5 receptor antagonists: Reduced human ether-a-go-go related gene potassium channel binding affinity and potent antiobesity effect
2009
Journal of Medicinal Chemistry
Nagaaki Sato
Makoto Ando
Shiho Ishikawa
Makoto Jitsuoka
Keita Nagai
Hirobumi Takahashi
Aya Sakuraba
Hiroyasu Tsuge
Hidefumi Kitazawa
Hisashi Iwaasa
Satoshi Mashiko
Akira Gomori
Ryuichi Moriya
Naoko Fujino
Tomoyuki Ohe
Akane Ishihara
Akio Kanatani
Takehiro Fukami
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Citations (22)
Discovery of substituted 2,4,4-triarylimidazoline derivatives as potent and selective neuropeptide Y Y5 receptor antagonists.
2009
Bioorganic & Medicinal Chemistry Letters
Nagaaki Sato
Makoto Jitsuoka
Shiho Ishikawa
Keita Nagai
Hiroyasu Tsuge
Makoto Ando
Osamu Okamoto
Hisashi Iwaasa
Akira Gomori
Akane Ishihara
Akio Kanatani
Takehiro Fukami
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Citations (13)
1