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Andrew Fisher
Andrew Fisher
Neurocrine Biosciences
Biochemistry
Chemistry
Chemical synthesis
Stereochemistry
Ligand (biochemistry)
5
Papers
72
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Synthesis and structure-activity relationships of spirohydantoin-derived small-molecule antagonists of the melanin-concentrating hormone receptor-1 (MCH-R1).
2007
Bioorganic & Medicinal Chemistry Letters
Martin W. Rowbottom
Troy Vickers
Junko Tamiya
Mingzhu Zhang
Brian Dyck
Jonathan Grey
David Schwarz
Christopher E. Heise
Michael Hedrick
Jenny Wen
Hui Tang
Hua Wang
Andrew Fisher
Anna Aparicio
John Saunders
Val S. Goodfellow
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Citations (8)
Synthesis and structure-activity relationships of retro bis- aminopyrrolidine urea (rAPU) derived small-molecule antagonists of the melanin-concentrating hormone receptor-1 (MCH-R1). Part 1
2006
Bioorganic & Medicinal Chemistry Letters
Martin W. Rowbottom
Troy Vickers
Brian Dyck
Jonathan Grey
Junko Tamiya
Mingzhu Zhang
Mehrak Kiankarimi
Dongpei Wu
Wesley Dwight
Warren Wade
David Schwarz
Christopher E. Heise
Ajay Madan
Andrew Fisher
Robert E. Petroski
Val S. Goodfellow
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Citations (6)
Synthesis and structure–activity relationships of uracil derived human GnRH receptor antagonists: (R)-3-[2-(2-amino)phenethyl]-1-(2,6-difluorobenzyl)-6-methyluracils containing a substituted thiophene or thiazole at C-5
2004
Bioorganic & Medicinal Chemistry Letters
Martin W. Rowbottom
Fabio C. Tucci
Patrick J. Connors
Timothy D. Gross
Yun-Fei Zhu
Zhiqiang Guo
Manisha Moorjani
Oscar Acevedo
Lee Carter
Susan K. Sullivan
Qiu Xie
Andrew Fisher
R. Scott Struthers
John Saunders
Chen Chen
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Citations (15)
3-(2-aminoalkyl)-1-(2,6-difluorobenzyl)-5- (2-fluoro-3-methoxyphenyl)-6-methyl-uracils as orally bioavailable antagonists of the human gonadotropin releasing hormone receptor.
2004
Journal of Medicinal Chemistry
Fabio C. Tucci
Yun-Fei Zhu
Zhiqiang Guo
Timothy D. Gross
Patrick J. Connors
Yinghong Gao
Martin W. Rowbottom
Struthers Rs
Greg J. Reinhart
Qiu Xie
Takung Chen
Haig Bozigian
Killam Bonneville Al
Andrew Fisher
L. Jin
John Saunders
Chen Chen
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Citations (29)
1