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Garret P. Textor
Garret P. Textor
Enzyme
Biochemistry
Chemistry
Tau-protein kinase
Lipophilicity
2
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123
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Discovery of a Tetrahydropyrimidin-2(1H)-one Derivative (TAK-442) as a Potent, Selective, and Orally Active Factor Xa Inhibitor
2010
Journal of Medicinal Chemistry
Takuya Fujimoto
Yasuhiro Imaeda
Noriko Konishi
Katsuhiko Hiroe
Masaki Kawamura
Garret P. Textor
Kathleen Aertgeerts
Keiji Kubo
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Citations (35)
2-{3-[4-(Alkylsulfinyl)phenyl]-1-benzofuran-5-yl}-5-methyl-1,3,4-oxadiazole derivatives as novel inhibitors of glycogen synthase kinase-3beta with good brain permeability.
2009
Journal of Medicinal Chemistry
Morihisa Saitoh
Jun Kunitomo
Eiji Kimura
Hiroki Iwashita
Yumiko Uno
Tomohiro Onishi
Noriko Uchiyama
Tomohiro Kawamoto
Toshimasa Tanaka
Clifford D. Mol
Douglas R. Dougan
Garret P. Textor
Gyorgy Snell
Masayuki Takizawa
Fumio Itoh
Masakuni Kori
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Citations (88)
1