Combined BCL-2 and HDAC Targeting Has Potent and TP53 Independent Activity In AML
Jessica M. SalmonGiovanna PomilioDonia MoujalledSarah MacRaildCharis E. TehSewa RijalAdam IveyTse-Chieh TehPaul G. EkertMarie SchoumacherLaurence Kraus‐BerthierIoana KloosDaniel H.D. GrayAndrew H. Wei
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Keywords:
Panobinostat
Venetoclax
Histone deacetylase inhibitor
<p>The top 35 genes most dramatically down-regulated by JQ1 and panobinostat combination therapy.</p>
Panobinostat
Histone deacetylase inhibitor
Histone deacetylase 2
HDAC8
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<p>The BET bromodomain proteins BRD3 and BRD4 induce N-Myc expression, but do not function synergistically.</p>
Panobinostat
BRD4
Histone deacetylase inhibitor
BET inhibitor
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<p>Combination therapy with JQ1 and panobinostat synergistically reduces neuroblastoma cell viability.</p>
Panobinostat
Histone deacetylase inhibitor
Vorinostat
HDAC11
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<p>JQ1 and panobinostat do not cooperatively induce apoptosis in normal non-malignant cells.</p>
Panobinostat
Histone deacetylase inhibitor
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<p>Combination therapy with JQ1 and panobinostat exerts synergistic anticancer effects in neuroblastoma cells.</p>
Panobinostat
Histone deacetylase inhibitor
Histone deacetylase 2
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<p>The BET bromodomain proteins BRD3 and BRD4 induce N-Myc expression, but do not function synergistically.</p>
BRD4
Panobinostat
Histone deacetylase inhibitor
BET inhibitor
Cite
Citations (0)
<p>JQ1 and panobinostat do not cooperatively induce apoptosis in normal non-malignant cells.</p>
Panobinostat
Histone deacetylase inhibitor
HDAC11
Cite
Citations (0)
<p>Combination therapy with JQ1 and panobinostat exerts synergistic anticancer effects in neuroblastoma cells.</p>
Panobinostat
Histone deacetylase inhibitor
Cite
Citations (0)
<p>JQ1 and panobinostat synergistically modulate gene expression.</p>
Panobinostat
Histone deacetylase inhibitor
Vorinostat
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Citations (0)
<p>The BET bromodomain protein BRD2 does not regulate N-Myc expression.</p>
Panobinostat
Histone deacetylase inhibitor
Cite
Citations (0)