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    Pyrano-[2,3b]-pyridines as potassium channel antagonists
    Bioorganic & Medicinal Chemistry Letters (2008)
    Heather J. FinlayJohn LloydMichael C. NymanMary Lee ConderTonya West
    Amide
    Carboxamide
    Potassium channel blocker
    Citations (15)
    Synthesis of amide isosteres of schweinfurthin-based stilbenes
    Bioorganic & Medicinal Chemistry (2017)
    David P. StockdaleJohn A. BeutlerDavid F. Wiemer
    Amide
    Carboxamide
    Citations (11)
    Synthesis and cytotoxicity of thieno[2,3-b]quinoline-2-carboxamide and cycloalkyl[b]thieno[3,2-e]pyridine-2-carboxamide derivatives
    Bioorganic & Medicinal Chemistry (2016)
    Euphemia LeungLisa I. PilkingtonMichelle van RensburgChae Yeon JeonMirae Song
    Quinoline
    Carboxamide
    IC50
    Citations (19)
    Synthesis and influenza virus sialidase inhibitory activity of analogues of 4-guanidino-Neu5Ac2en (GG167) with modified 5-substituents
    European Journal of Medicinal Chemistry (1996)
    PW SmithI. D. STARKEYP. D. HOWESS. L. SOLLISSP Keeling
    Sialidase
    Structure–activity relationship
    Carboxamide
    Amide
    Sulfonamide
    Influenzavirus B
    Pyran
    Citations (50)
    Pyridine amides as potent and selective inhibitors of 11β-hydroxysteroid dehydrogenase type 1
    Bioorganic & Medicinal Chemistry Letters (2008)
    Haixia WangZheming RuanJames J. LiLigaya M. SimpkinsRebecca A. Smirk
    Amide
    Carboxamide
    Structure–activity relationship
    Citations (22)
    Synthesis and evaluation of two series of 4′-aza-carbocyclic nucleosides as adenosine A2A receptor agonists
    Bioorganic & Medicinal Chemistry Letters (2009)
    David T. BeattieAndrew BrearleyZarin BrownSteven J. CharltonBrian J. Cox
    Carboxamide
    Amide
    Citations (10)
    Structure–activity relationship studies of manzamine A: Amidation of positions 6 and 8 of the β-carboline moiety
    Bioorganic & Medicinal Chemistry (2009)
    Amir E. WahbaJiangnan PengSucheta KudrimotiBabu L. TekwaniMark T. Hamann
    Amide
    Carboxamide
    Structure–activity relationship
    Plasmodium berghei
    Moiety
    Citations (25)
    1,4-Diacylpiperazine-2-(S)-[(N-aminoalkyl)carboxamides] as novel, potent substance P receptor antagonists.
    Bioorganic & Medicinal Chemistry Letters (1993)
    Sander G. MillsMu Tsu WuMalcolm MacCossRichard J. BudhuConrad P. Dorn
    Carboxamide
    Amide
    Citations (13)
    Stereoselective synthesis and biological evaluation of 3,4-diaminocyclohexanecarboxylic acid derivatives as factor Xa inhibitors
    Bioorganic & Medicinal Chemistry Letters (2008)
    Tsutomu NagataMasatoshi NagamochiShozo KobayashiSatoshi KomoriyaToshiharu Yoshino
    Amide
    Carboxamide
    Hydroxamic acid
    Citations (17)
    Oxadiazoles as bioisosteric transformations of carboxylic functionalities. II
    European Journal of Medicinal Chemistry (1996)
    Knud Erik AndersenB. F. LUNDTA.S. JørgensenC. Bræstrup
    Amide
    Moiety
    Carboxamide
    Oxadiazole
    Citations (79)