Diversity Oriented Synthesis: Substitution at C5 in Unreactive Pyrimidines by Claisen Rearrangement and Reactivity in Nucleophilic Substitution at C2 and C4 in Pteridines and Pyrido[2,3‐d]pyrimidines.

2011 
A number of diversified pyridopyrimidines and pteridines are prepared and their biological activity is screened.
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