The effect of macrocyclic chelators on the targeting properties of the 68Ga-labeled gastrin releasing peptide receptor antagonist PEG2-RM26

Zohreh Varasteh,Bogdan Mitran,Ulrika Rosenström,Irina Velikyan,Maria Rosestedt,Gunnar Lindeberg,Jens Nørkær Sørensen,Mats Larhed,Vladimir Tolmachev,Anna Orlova

The effect of macrocyclic chelators on the targeting properties of the 68Ga-labeled gastrin releasing peptide receptor antagonist PEG2-RM26

2015

Zohreh Varasteh
Bogdan Mitran
Ulrika Rosenström
Irina Velikyan
Maria Rosestedt
Gunnar Lindeberg
Jens Nørkær Sørensen
Mats Larhed
Vladimir Tolmachev
Anna Orlova

INTRODUCTION: Overexpression of gastrin-releasing peptide receptors (GRPR) has been reported in several cancers. Bombesin (BN) analogs are short peptides with a high affinity for GRPR. Different BN ...

Keywords:

DOTA
Biochemistry
Gastrin-releasing peptide receptor
Bombesin
Peptide
Receptor
Chemistry
Antagonist

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