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Phenethanolamines and their uses

1984 
ON PREPARE NEW COMPOSITIONS USING AGONISTS B SPECIAL AND MATERIALS vehicular AND ARE USEFUL FOR PRODUCTION OF ANTI-INFLAMMATORY TOPICAL MAMMALS. THE AGONIST B SELECTED WERE NOT KNOWN IN ADVANCE TO PRESENT ANTI-INFLAMMATORY ACTIVITY TOPICAL. COMPOSITIONS APPLIED FOR EXAMPLE IN THE FORM OF SPRAYING, BAUMES, CREAMS, GELS, LOTIONS, AND SUPPOSITORIES ALL TO BE APPLIED TO MAMMALS SO TOPICAL VS. SYSTEMIC A. THE N- (3 indolyl-ISOPROPYL) - AND N- (3-iNDOLYL-T-butyl) -2- (4-HYDROXY-3-methanesulfonamidophenyl) -2-hydroxyethylamines PHARMACEUTICALLY ACCEPTABLE AND THEIR SALTS ARE ANTI-ASTHMA AND THE SHOWS bronchodilator THEIR ACTION AND INHIBITION OF SMOOTH MUSCLE CONTRACTION CAUSED BY THE RELEASE INDUCED BY ANTIGEN OF CHEMICAL MEDIATORS.
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