Enantioselective Organocatalytic Synthesis of Oxazolidine Derivatives through a One‐Pot Cascade Reaction

An asymmetric organocatalytic cascade reaction which can afford a series of oxazolidine derivatives has been developed. The one-pot reaction reported here can produce an oxazolidine derivative in a highly enantioselective manner and good yield with good to excellent diastereomeric ratio.