UNIT 1.26 Characterization of Cannabinoid Receptors

This unit describes the use of cannabinoid radioligands in competitive binding assays for determining affinity parameters (IC50, Ki) of unlabeled compounds at transfected CB1 and CB2 receptors expressed in cell lines. Curr. Protoc. Pharmacol. 63:1.26.1-1.26.10. © 2013 by John Wiley & Sons, Inc. Keywords: cannabinoids; receptor binding; GPR 55