Synthesis of Alkyl Hexahydropyrazino[1,2‐c]pyrimidine‐9‐carboxylates

2012 
via cyclocondensation of 3-alkoxycarbonylmethylidenepiperazinones (I) with α-chlorobenzyl isocyanates or 1-aryl-2,2,2-trifluoroethyl isocyanates
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