Facile Preparation and Suzuki—Miyaura Cross-Coupling of N-2-Alkylated 2H-1,2,3-Triazole 4-Boronates.

A novel protocol is developed to prepare 2H-1,2,3-triazoles, functionalized with a boronate moiety at C-4 such as the pharmaceutically important system (VI) and its Thp analogue (IX).