Allophenylnorstatine containing HIV-1 protease inhibitors: design, synthesis and structure-activity relationships for selected P2 ligands

1999 
ﻊﻗﻮﻣﺮﻴﻴﻐﺗو ﻦﻴﻣأ ﻞﻳﺰﻨﺑ ﻞﻴﺜﻴﻣ وا ﻦﻴﻣأ ﻞﻴﺗﻮﻴﺑ ﻰﺛﻼﺜآ ﻢﺗو لﻮﻣوﺮﻜﻴﻣ 5 ىﻮﺘﺴﻣ ﺪﻨﻋ ﻢﻳﺰﻧﻻا ﻂﻴﺒﺜﺘﻟ ﺔﻳﻮﺌﻣ ﺔﺒﺴﻨآ ﺔﻘﻠﺨﻤﻟا تﺎﺒآﺮﻤﻟا ﻩﺬه ﺔﻴﻠﻋﺎﻔﻟ ﻰﺋﺪﺒﻤﻟا ﻢﻴﻴﻘﺘﻟا ﺐﺒﺴﻤﻟا سوﺮﻴﻔﻟا ﻰﻓ ﺰﻴﻴﺗوﺮﺒﻟا ﻢﻳﺰﻧﻻ تﺎﻄﺒﺜﻤآ ﺔﻴﻠﻋﺎﻔﻟاو ﻰﺋﺎﻴﻤﻴﻜﻟا ﺐﻴآﺮﺘﻟا ﻦﻴﺑ ﻰﻠﺜﻤﻟا ﺔﻗﻼﻌﻟا ﺔﺳارد ﻞﻳﺰﻨﺑ ﻞﻴﺜﻴﻣ-2 ﻰﻠﻋ ﺔﻳﻮﺘﺤﻤﻟا تﺎﺒآﺮﻤﻟا نا ﺞﺋﺎﺘﻨﻟا ﺖﺘﺒﺛا .ﻪﺑ ةﺮﺛﺆﻤﻟا تﺎﻋﻮﻤﺠﻤﻟاو ﻰﻣدﻻا ﺔﻋﺎﻨﻤﻟا ﺺﻘﻨﻟ
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