Synthesis of 5,7-Dichloro-6-azaindolesand Functionalization via a Highly Selective Lithium-Chlorine Exchange
2009
The synthesis of a range of novel 5,7-dichloro-6-azaindoles through the use of a Fischer cyclization with pyridine hydrochloride in N-methylpyrrolidin-2-one is described. Dichloro-6-azaindoles are versatile compounds that can be selectively substituted through a palladium-catalyzed cross-coupling reaction or a high-yielding lithium-chlorine exchange.
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