A Palladium‐Catalyzed Domino Approach to 2,3‐Disubstituted Benzofurans via an Intermolecular Carbopalladation/C(sp3)−H Functionalization/Isomerization Sequence

A palladium-catalyzed domino strategy has been developed for the synthesis of 2,3-disubstituted benzofuran derivatives. This cascade reaction sequence involves intermolecular carbopalladation and C(sp3)−H functionalization followed by isomerization.