Synthesis and SAR of amino acid-derived heterocyclic progesterone receptor full and partial agonists
2009
Abstract Two classes of amino acid-derived heterocyclic progesterone receptor ligands were developed to address the metabolic issues posed by the dimethyl amide functionality of the lead compound ( 1) . The tetrazole-derived ligands behaved as potent partial agonists, while the 1,2,4-triazole ligands behaved as potent full agonists.
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