Azide–Enolate 1,3‐Dipolar Cycloaddition as an Efficient Approach for the Synthesis of 1,5‐Disubstituted 1,2,3‐Triazoles from Alkyl/Aryl Azides and β‐Ketophosphonates

Davir González-Calderón,Aydeé Fuentes-Benítes,Eduardo Díaz-Torres,Carlos A. González-González,Carlos González-Romero

Azide–Enolate 1,3‐Dipolar Cycloaddition as an Efficient Approach for the Synthesis of 1,5‐Disubstituted 1,2,3‐Triazoles from Alkyl/Aryl Azides and β‐Ketophosphonates

2016

Davir González-Calderón
Aydeé Fuentes-Benítes
Eduardo Díaz-Torres
Carlos A. González-González
Carlos González-Romero

A simple procedure to prepare 1,5-disubstituted 1,2,3-triazoles efficiently from alkyl/aryl azides and β-ketophosphonates in the presence of KOH by an azide–enolate 1,3-dipolar cycloaddition in good yields was developed.

Keywords:

Photochemistry
Organic chemistry
Chemistry
1,3-Dipolar cycloaddition
Aryl
Alkyl
Cycloaddition
Azide

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