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Jesse Brodkin
Jesse Brodkin
General Atomics
Metabotropic glutamate receptor 5
Antagonist
MTEP
Biochemistry
Metabotropic glutamate receptor
8
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929
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0.01
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Discovery of novel modulators of metabotropic glutamate receptor subtype-5.
2004
Bioorganic & Medicinal Chemistry
Bowei Wang
Jean-Michel Vernier
Sara Rao
Janice Chung
Jeffery J. Anderson
Jesse Brodkin
Xiaohui Jiang
Michael F. Gardner
Xiaoqing Yang
Benito Munoz
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Citations (29)
Discovery of Novel Heteroarylazoles That Are Metabotropic Glutamate Subtype 5 Receptor Antagonists with Anxiolytic Activity
2004
Journal of Medicinal Chemistry
Jeffrey Roger Roppe
Nicholas D. Smith
Dehua Huang
Lida Tehrani
Bowei Wang
Jeffrey Anderson
Jesse Brodkin
Janice Chung
Xiaohui Jiang
Christopher King
Benito Munoz
Mark A. Varney
Petpiboon Prasit
Nicholas D. P. Cosford
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Citations (116)
3-[(2-Methyl-1,3-thiazol-4-yl)ethynyl]-pyridine: a potent and highly selective metabotropic glutamate subtype 5 receptor antagonist with anxiolytic activity.
2003
Journal of Medicinal Chemistry
Nicholas D. P. Cosford
Lida Tehrani
Jeffrey Roger Roppe
Edwin J. Schweiger
Nicholas D. Smith
Jeffrey Anderson
Linda J. Bristow
Jesse Brodkin
Xiaohui Jiang
Ian A. McDonald
Sara Rao
Mark S. Washburn
Mark A. Varney
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Citations (380)
Anxiolytic-like activity of the mGluR5 antagonist MPEP: A comparison with diazepam and buspirone
2002
Pharmacology, Biochemistry and Behavior
Jesse Brodkin
Chris S. Busse
Stacey J Sukoff
Mark A. Varney
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Citations (136)
Reduced stress-induced hyperthermia in mGluR5 knockout mice
2002
European Journal of Neuroscience
Jesse Brodkin
M. Bradbury
Chris S. Busse
N. Warren
L. J. Bristow
Mark A. Varney
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Citations (71)
1