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Scott Lamont

AstraZeneca

31

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876

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Tricyclic Indazoles—A Novel Class of Selective Estrogen Receptor Degrader Antagonists

2019 Journal of Medicinal Chemistry
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An investigation into the role of 2,6-lutidine as an additive for the RuCl3-NaIO4 mediated oxidative cleavage of olefins to ketones

2018 Tetrahedron Letters
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Structure-Guided Discovery of Potent and Selective Inhibitors of ERK1/2 from a Modestly Active and Promiscuous Chemical Start Point.

2017 Journal of Medicinal Chemistry
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Optimization of a Series of Bivalent Triazolopyridazine Based Bromodomain and Extraterminal Inhibitors: The Discovery of (3R)-4-[2-[4-[1-(3-Methoxy-[1,2,4]triazolo[4,3-b]pyridazin-6-yl)-4-piperidyl]phenoxy]ethyl]-1,3-dimethyl-piperazin-2-one (AZD5153)

2016 Journal of Medicinal Chemistry
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Discovery of 4,6-disubstituted pyrimidines as potent inhibitors of the heat shock factor 1 (HSF1) stress pathway and CDK9 (vol 7, pg 1580, 2016)

2016
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Discovery and Characterization of MAPK-activated Protein Kinase-2 Prevention of Activation Inhibitors

2015 Journal of Medicinal Chemistry
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Structure-Based Design of Potent and Selective Inhibitors of the Metabolic Kinase PFKFB3

2015 Journal of Medicinal Chemistry
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Optimization of a Novel Binding Motif to (E)-3-(3,5-Difluoro-4-((1R,3R)-2-(2-Fluoro-2-Methylpropyl)-3-Methyl-2, 3,4,9-Tetrahydro-1H-Pyrido[3,4-B]Indol-1-Yl)Phenyl)Acrylic Acid (Azd9496), a Potent and Orally Bioavailable Selective Estrogen Receptor Downregulator and Antagonist.

2015 Journal of Medicinal Chemistry
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Regioselective ortho alkylation of nitro indole, carbazole, benzothiophene and benzofuran

2015 Tetrahedron Letters
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Discovery of a Potent and Selective EGFR Inhibitor (AZD9291) of Both Sensitizing and T790M Resistance Mutations That Spares the Wild Type Form of the Receptor

2014 Journal of Medicinal Chemistry
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Citations (327)