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Andreas Mühlemann
Andreas Mühlemann
Hoffmann-La Roche
Chemistry
Receptor
Metabotropic receptor
Allosteric regulation
Biochemistry
5
Papers
457
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Determination of key amino acids implicated in the actions of allosteric modulation by 3,3'-difluorobenzaldazine on rat mGlu5 receptors.
2006
European Journal of Pharmacology
Andreas Mühlemann
Natalie A. Ward
Nicole A. Kratochwil
Catherine Diener
Christophe Fischer
Andy Stucki
Georg Jaeschke
Pari Malherbe
Richard Hugh Philip Porter
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Citations (56)
An automated system for the analysis of G protein-coupled receptor transmembrane binding pockets: alignment, receptor-based pharmacophores, and their application.
2005
Journal of Chemical Information and Modeling
Nicole A. Kratochwil
Pari Malherbe
Lothar Lindemann
Martin Ebeling
Marius C. Hoener
Andreas Mühlemann
Richard Hugh Philip Porter
Martin Stahl
Paul R. Gerber
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Citations (58)
Fenobam: A Clinically Validated Nonbenzodiazepine Anxiolytic Is a Potent, Selective, and Noncompetitive mGlu5 Receptor Antagonist with Inverse Agonist Activity
2005
Journal of Pharmacology and Experimental Therapeutics
Richard Hugh Philip Porter
Georg Jaeschke
Will Spooren
Theresa M. Ballard
Bernd Büttelmann
Sabine Kolczewski
Jens-Uwe Peters
Eric Prinssen
Jürgen Wichmann
Eric Vieira
Andreas Mühlemann
Silvia Gatti
Vincent Mutel
Pari Malherbe
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Citations (272)
Constitutive activity modulation of human metabotropic glutamate 5a receptors in HEK293 cells: a role for key amino‐terminal cysteine residues
2005
British Journal of Pharmacology
Andreas Mühlemann
Catherine Diener
Christophe Fischer
Jenny Piussi
Andy Stucki
Richard Hugh Philip Porter
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Citations (6)
1